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Comparative Protein Binding of Diazepam and Desmethyldiazepam

โœ Scribed by ALLEN, MARCIA DIVOLL; GREENBLATT, DAVID J.


Book ID
121430762
Publisher
Sage Publications
Year
1980
Tongue
English
Weight
507 KB
Volume
20
Category
Article
ISSN
0091-2700

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๐Ÿ“œ SIMILAR VOLUMES


Binding of diazepam and desmethyldiazepa
โœ Marcia Divoll; David J. Greenblatt ๐Ÿ“‚ Article ๐Ÿ“… 1981 ๐Ÿ› Springer ๐ŸŒ English โš– 279 KB

The binding of diazepam (DZ) and its major metabolite desmethyldiazepam (DMDZ) to plasma protein was evaluated in a series of controlled in vitro studies using equilibrium dialysis. Free fraction (FF) of both drugs alone changed significantly with total plasma drug concentration, but the increased F