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ChemInform Abstract: Synthesis of Phenoxyacetic Acid Derivatives as Highly Potent Antagonists of Gastrin/Cholecystokinin-B Receptors. Part 2.

✍ Scribed by Y. TAKEDA; ET AL. ET AL.

Publisher: John Wiley and Sons
Year: 2010
Weight: 30 KB
Volume: 29
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.199847292

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✦ Synopsis

Synthesis of Phenoxyacetic Acid Derivatives as Highly Potent Antagonists of Gastrin/Cholecystokinin-B Receptors. Part 2.

-In order to increase the potency and selectivity as gastrin antagonists of recently obtained structures a novel series of compounds such as (I) is synthesized. The most potent compounds are (II). Thus, (IIa) shows similar antisecretory activity to YM022 when administered intraduodenally. -(TAKEDA, Y.

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