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ChemInform Abstract: Synthesis of N1-Substituted Analogues of (2R,4R)-4-Aminopyrrolidine-2,4-dicarboxylic Acid as Agonists, Partial Agonists, and Antagonists of Group II Metabotropic Glutamate Receptors.

✍ Scribed by Jayanta Kumar Mukhopadhyaya; Alan P. Kozikowski; Ewa Grajkowska; Sergey Pshenichkin; Jarda T. Wroblewski

Publisher: John Wiley and Sons
Year: 2010
Weight: 34 KB
Volume: 32
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.200145201

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ChemInform Abstract: Spiro-Substituted P

ChemInform Abstract: Spiro-Substituted Piperidines as Neurokinin Receptor Antagonists. Part 3. Synthesis of (.+-.)-N-[2-(3,4-Dichlorophenyl)-4-(spiro-substituted piperidin-1′-yl)butyl]-N-methylbenzamides and Evaluation of NK1—NK2 Dual Antagonistic Activities.

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ChemInform Abstract: Methylated Analogue

ChemInform Abstract: Methylated Analogues of Methyl (R)-4-(3,4-Dichlorophenylacetyl)-3- (pyrrolidin-1-ylmethyl)piperazine-1-carboxylate (GR-89,696) as Highly Potent ϰ-Receptor Agonists: Stereoselective Synthesis, Opioid-Receptor Affinity, Receptor Selectivity, and Functional Studies.

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## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable v

ChemInform Abstract: Spiro-Substituted P

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