ChemInform Abstract: Synthesis and hSERT Activity of Homotryptamine Analogues. Part 6. [3 + 2] Dipolar Cycloaddition of 3-Vinylindoles.
β Scribed by Lawrence R. Marcin; Ronald J. Mattson; Qi Gao; Dedong Wu; Thaddeus F. Molski; Gail K. Mattson; Nicholas J. Lodge
- Publisher
- John Wiley and Sons
- Year
- 2010
- Weight
- 23 KB
- Volume
- 41
- Category
- Article
- ISSN
- 0931-7597
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β¦ Synopsis
Abstract
A series of homotryptamine analogues such as (V) and (VIII) is prepared via [3 + 2] dipolar cycloaddition of vinylindole (I) with cyclic nitrones as key step.
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