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ChemInform Abstract: Synthesis and Evaluation of Highly Potent GABAA Receptor Antagonists Based on Gabazine (SR-95531).

✍ Scribed by Favaad Iqbal; Ryan Ellwood; Martin Mortensen; Trevor G. Smart; James R. Baker

Publisher: John Wiley and Sons
Year: 2011
Weight: 34 KB
Volume: 42
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.201148169

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✦ Synopsis

Abstract

The compounds (VIa) and (VII) are highly potent GABA~A~ receptor antagonists compared to the parent antagonist gabazine.

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