𝔖 Bobbio Scriptorium
✦   LIBER   ✦

ChemInform Abstract: Stereoselective Conjugate Addition Directed by an Enantiomerically Pure Ketal. Preparation of the Cyclohexanone Fragment of N-Methylwelwitindolinone C Isothiocyanate.

✍ Scribed by J. P. KONOPELSKI; H. DENG; K. SCHIEMANN; J. M. KEANE; M. M. OLMSTEAD


Publisher
John Wiley and Sons
Year
2010
Weight
32 KB
Volume
30
Category
Article
ISSN
0931-7597

No coin nor oath required. For personal study only.

✦ Synopsis


Stereoselective Conjugate Addition Directed by an Enantiomerically Pure Ketal. Preparation of the Cyclohexanone Fragment of N-Methylwelwitindolinone C Isothiocyanate.

-A cyclohexanone intermediate (V), which may be employed in the synthesis of the marine natural product N-methylwelwitindolinone C isothiocyanate, is prepared based on a diastereoselective conjugate addition of Grignard reagent (II) to the α,β-unsaturated ketone (I) bearing an adjacent chiral ketal as directing group.

-(KONOPELSKI,