𝔖 Bobbio Scriptorium
✦   LIBER   ✦

ChemInform Abstract: Probing the Importance of Spacial and Conformational Domains in Captopril Analogues for Angiotensin Converting Enzyme Activity.

✍ Scribed by S. HANESSIAN; U. REINHOLD; M. SAULNIER; S. CLARIDGE


Publisher
John Wiley and Sons
Year
2010
Weight
29 KB
Volume
30
Category
Article
ISSN
0931-7597

No coin nor oath required. For personal study only.

✦ Synopsis


Probing the Importance of Spacial and Conformational Domains in Captopril Analogues for Angiotensin Converting Enzyme Activity.

-An improved large-scale synthesis of 4,5-methano-prolines (IV) and (V) and the enzymatic activity of the corresponding N-(3-mercapto-2-methyl-propionyl) derivatives, e.g. (VIII), as ACE-inhibitors is described. -(HANESSIAN, S.;