Optimization of the Suzuki coupling reac
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Marija Alešković; Nikola Basarić; Kata Mlinarić-Majerski
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Article
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2011
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Journal of Heterocyclic Chemistry
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English
⚖ 233 KB
## Abstract A facile three‐step synthesis of 2‐(2‐aminophenyl)pyrrole (**1**) and 2‐[(2‐aminomethyl)phenyl]pyrrole (**2**) is reported by use of Suzuki coupling of __N__‐Boc‐pyrrol‐2‐yl boronic acid (**3**) and o‐substituted aryl halogenides, followed by hydrogenation. The Pd‐catalyzed cross‐coupli