ChemInform Abstract: One-Pot Synthesis of Pyrimido[1,6-a]indol-1(2H)-one Derivatives by a Nucleophilic Addition/Cu-Catalyzed N-Arylation/Pd-Catalyzed C—H Activation Sequential Process.

✍ Scribed by Zhi-Jing Wang; Jian-Guo Yang; Fan Yang; Weiliang Bao

• Publisher: John Wiley and Sons
• Year: 2010
• Weight: 48 KB
• Volume: 41
• Category: Article
• ISSN: 0931-7597
• DOI: 10.1002/chin.201046161

✦ Synopsis

Abstract

The reaction is applicable to a variety of ortho‐gem‐dibromovinyl isocyanates and N‐alkyl anilines and tolerates substitution at all positions on the aromatic rings.