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ChemInform Abstract: Novel Imidazobenzazepine Derivatives as Dual H1/5-HT2A Antagonists for the Treatment of Sleep Disorders.

✍ Scribed by Massimo Gianotti; Corrado Corti; Sonia Delle Fratte; Romano Di Fabio; Colin P. Leslie; Francesca Pavone; Laura Piccoli; Luigi Stasi; Mark J. Wigglesworth

Publisher: John Wiley and Sons
Year: 2010
Weight: 24 KB
Volume: 42
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.201101209

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✦ Synopsis

Abstract

The derivatives (I) are shown to possess potent and balanced H~1~/5‐HT~2A~ receptor antagonist activities.

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