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ChemInform Abstract: New Pyrrolobenzothiazepine Derivatives as Molecular Probes of the “ Peripheral-Type” Benzodiazepine Receptor (PBR) Binding Site.

✍ Scribed by G. CAMPIANI; V. NACCI; I. FIORINI; M. P. DE FILIPPIS; A. GAROFALO; S. M. CIANI; G. GRECO; E. NOVELLINO; C. MANZONI; T. MENNINI

Publisher: John Wiley and Sons
Year: 2010
Weight: 34 KB
Volume: 28
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.199733221

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✦ Synopsis

New Pyrrolobenzothiazepine Derivatives as Molecular Probes of the " Peripheral-Type" Benzodiazepine Receptor (PBR) Binding Site.

-A series of new pyrrolobenzothiazepine derivatives (VI) and a pyrrolobenzothiazocine derivative (X) are prepared and evaluated for their affinity towards the PBR. Compound (VId) is found to be the most potent ligand for this receptor in this series.

-(CAMPIANI, G.; NACCI, V.;

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