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ChemInform Abstract: Lipase PS (Pseudomonas cepacia) Mediated Resolution of β-Substituted γ-((Acetyloxy)methyl)-γ-butyrolactones: Complete Stereochemical Reversion by Substituents.

✍ Scribed by Hyung-Joon Ha; Kyung-Noh Yoon; Sang-Youn Lee; Young-Soo Park; Moon-Soo Lim; Yoon-Gil Yim


Publisher
John Wiley and Sons
Year
2010
Weight
33 KB
Volume
30
Category
Article
ISSN
0931-7597

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✦ Synopsis


Lipase PS (Pseudomonas cepacia) Mediated Resolution of β-Substituted γ-((Acetyloxy)methyl)-γ-butyrolactones: Complete Stereochemical Reversion by Substituents.

-The resolution of lactones (I), (III), and (V) with lipase PS proceeds with high selectivity and reversal of the stereochemical preference for cis-or trans-β-substituted lactones. Similar results are obtained for the corresponding cis and trans ethyl derivatives. Lactones with larger cis-or trans-β-substituents such as phenyl show almost no stereodifferentiation.