ChemInform Abstract: Enantioselective Organocatalytic Synthesis of Highly Functionalized Tetrahydrothiophenes by a Michael-Aldol Cascade Reaction.
β Scribed by Guangshun Luo; Shilei Zhang; Wenhu Duan; Wei Wang
- Publisher
- John Wiley and Sons
- Year
- 2009
- Weight
- 26 KB
- Volume
- 40
- Category
- Article
- ISSN
- 0931-7597
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Highly Enantioselective Organocatalytic Cascade Reaction for the Synthesis of Piperidines and Oxazolidines. -Organocatalyzed Michael addition of amidomalonates, e.g. (I) and (VI), towards enals (II) followed by intramolecular hemiaminal formation provides enantioenriched piperidine derivatives (III)
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