ChemInform Abstract: Efficient Two-Step Syntheses of Sulfonylguanidines from Sulfonamides.
β Scribed by P. DEPREZ; J.-P. VEVERT
- Publisher
- John Wiley and Sons
- Year
- 2010
- Weight
- 29 KB
- Volume
- 28
- Category
- Article
- ISSN
- 0931-7597
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β¦ Synopsis
The title sulfonylguanidines (V) or (IX), potent bioisosteres of the tetrazole moiety common to most of the AII antagonists under development, are prepared on two routes with moderate to good yields.
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