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ChemInform Abstract: (E)-3-(2-(N-Phenylcarbamoyl)vinyl)pyrrole-2-carboxylic Acid Derivatives. A Novel Class of Glycine Site Antagonists.

✍ Scribed by G. TARZIA; ET AL. ET AL.

Publisher: John Wiley and Sons
Year: 2010
Weight: 32 KB
Volume: 29
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.199827131

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✦ Synopsis

27 -131

(E)-3-(2-(N-Phenylcarbamoyl)vinyl)pyrrole-2-carboxylic Acid Derivatives. A Novel Class of Glycine Site Antagonists.

-A series of the title compounds is evaluated for in vitro affinity at the strychnine-insensitive glycine-binding site of the N-methyl-D-aspartate receptor complex. The most active compounds are (IVa), (IVb), and (VII). -(TARZIA, G.; ET AL.; J.

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