Selective difluorination, introducing a lactame moiety (instead of an amine) and a double bond in a trihydroxy-2-thiaquinolizidine derivative reverses the selectivity of the glycosidase inhibitor -a selective inhibitor for an a-glucosidase is altered into an excellent, competitive inhibitor for a bg
ChemInform Abstract: Difluorotetrahydropyridothiazinone: A Selective β-Galactosidase Inhibitor.
✍ Scribed by Rene Csuk; Erik Prell
- Publisher
- John Wiley and Sons
- Year
- 2011
- Weight
- 29 KB
- Volume
- 42
- Category
- Article
- ISSN
- 0931-7597
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