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ChemInform Abstract: Development of Bioactive Functions in Hydrangeae Dulcis Folium. Part 6. Syntheses of Thunberginols A and F and Their 3′-Deoxy-Derivatives Using Regiospecific Lactonization of Stilbene Carboxylic Acid: Structures and Inhibitory Activity on Histamine Release of Hydramacrophyllols A and B.

✍ Scribed by M. YOSHIKAWA; H. SHIMADA; N. YAGI; N. MURAKAMI; H. SHIMODA; J. YAMAHARA; H. MATSUDA


Publisher
John Wiley and Sons
Year
2010
Weight
36 KB
Volume
28
Category
Article
ISSN
0931-7597

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✦ Synopsis


Development of Bioactive Functions in Hydrangeae Dulcis Folium. Part 6. Syntheses of Thunberginols A and F and Their 3'-Deoxy-Derivatives Using Regiospecific Lactonization of Stilbene Carboxylic Acid: Structures and Inhibitory Activity on Histamine Release of Hydramacrophyllols A and B.

-Thunberginol A (IV) and F (X) (constituents of Hydrangeae Dulcis Folium) and the corresponding 3'-deoxyderivatives (V) and (XI) are synthesized in order to study their antiallergic activity. Hydramacrophyllos A and B (cf. (XII)), isolated together with (IV) and (X), are found to inhibit the histamine release from rat peritoneal exudate cells induced by antigen-antibody reaction. -(YOSHIKAWA, M.;