ChemInform Abstract: Design, Synthesis, and Pharmacological Characterization of 4-[4,4-Dimethyl-3-(4-hydroxybutyl)-5-oxo-2-thioxo-1-imidazolidinyl] -2-iodobenzonitrile as a High-Affinity Nonsteroidal Androgen Receptor Ligand.

ChemInform Abstract: Design and Synthesi

ChemInform Abstract: Design and Synthesis of 4-[3,5-Dioxo-11-oxa-4,9-diazatricyclo [5.3.1.02,6]undec-4-yl]-2-trifluoromethyl-benzonitriles as Androgen Receptor Antagonists.

✍ Hai-Yun Xiao; et al. et al. 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 20 KB 👁 1 views

## Abstract Based on the common structure of androgen receptor (AR) antagonists, a series of novel diazatricyclic compounds is designed.

ChemInform Abstract: Synthesis and Biolo

ChemInform Abstract: Synthesis and Biological Evaluation of Novel 9-Heteroaryl Substituted 7-Chloro-4,5-dihydro-4-oxo-1,2,4-triazolo [1,5-a]quinoxaline-2-carboxylates (TQX) as (R,S)-2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid (AMPA) Receptor Antagonists.

✍ Daniela Catarzi; Vittoria Colotta; Flavia Varano; Guido Filacchioni; Paola Gratt 📂 Article 📅 2009 🏛 John Wiley and Sons ⚖ 45 KB 👁 1 views

ChemInform Abstract: Design, Synthesis,

ChemInform Abstract: Design, Synthesis, and Biological Evaluation of a Second Generation of Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as Potent and Selective A2A Adenosine Receptor Antagonists.

✍ P. G. BARALDI; B. CACCIARI; G. SPALLUTO; M. BERGONZONI; S. DIONISOTTI; E. ONGINI 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 43 KB 👁 2 views

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable v

Probes for narcotic receptor mediated ph

Probes for narcotic receptor mediated phenomena 22. (1) synthesis and characterization of optically pure [3H](+)-4-[(αR)-α-((2S, 5R)-4-propyl-2,5-dimethyl-1-piperazinyl)-3-methoxybenzyl]-N, N-diethylbenzamide, [3H]SNC 121, a novel high affinity and selective ligand for delta opioid receptors

✍ Silvia N. Calderon; Craig M. Bertha; J. Silvio Gutkind; Heng Xu; John S. Partill 📂 Article 📅 1996 🏛 John Wiley and Sons 🌐 French ⚖ 236 KB 👁 2 views

Probes for Narcotic Receptor Mediated Phenomena 22. (1) Synthesis and Characterization of Optically Pure [3 H I ( +)-4-1 ( a R)-a -( ( 2 s ,5 R ) -4 -P r o p y I -2 , 5 -d i m e t h y l -l -p i p e r e z i n y l ) -3 -m e t h o x y b e n z y l ] -~, ~-d i e t h y l b e n z a m i d e , [3H]SNC 121, a

ChemInform Abstract: 3-Amino-3,4-dihydro

ChemInform Abstract: 3-Amino-3,4-dihydro-2H-1-benzopyran Derivatives as 5-HT1A Receptor Ligands and Potential Anxiolytic Agents. Part 2. Synthesis and Quantitative Structure-Activity Relationship Studies of Spiro( pyrrolidine- and piperidine-2,3′(2′H)-benzopyrans).

✍ C. COMOY; C. MAROT; T. PODONA; M.-L. BAUDIN; L. MORIN-ALLORY; G. GUILLAUMET; B. 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 33 KB 👁 1 views

ChemInform Abstract: Studies on the Chem

ChemInform Abstract: Studies on the Chemistry of Thienoanellated O,N- and S,N-Containing Heterocycles. Part 22. Synthesis of 1,2,4-Oxadiazolylimidazo[1,5-a]thieno[2,3-e]pyrazines as Ligands for the γ-Aminobutyric Acid A/Benzodiazepine Receptor Complex.

✍ Thomas Erker; Karin Trinkl 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 33 KB 👁 2 views

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable v