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ChemInform Abstract: Biginelli Reaction Beyond Three-Component Limit: Synthesis of Functionalized Pyrimidinones via a One-Pot Biginelli-Pd Mediated C—C Coupling Strategy.

✍ Scribed by P. Mahesh Kumar; K. Siva Kumar; Srinivas Reddy Poreddy; Pradeep Kumar Mohakhud; K. Mukkanti; Manojit Pal

Publisher: John Wiley and Sons
Year: 2011
Weight: 54 KB
Volume: 42
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.201125163

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✦ Synopsis

Abstract

The synthesis of novel 3,4‐dihydropyrimidinone derivatives involves sequential H~3~PO~4~‐catalyzed solvent‐free Biginelli reaction followed by copper‐free Sonogashira, Heck or Suzuki coupling.

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