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ChemInform Abstract: Active Thionium Species Mediated Functionalization at the 2α-Position of Indole Derivatives.

✍ Scribed by Kazuhiro Higuchi; Masanori Tayu; Tomomi Kawasaki

Publisher: John Wiley and Sons
Year: 2011
Weight: 48 KB
Volume: 42
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.201142107

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✦ Synopsis

Abstract

The 2α‐functionalization of indole derivatives such as tetrahydrocarbazoles and the pyridoindole derivative (VII), a core structure of biologically active natural products, is achieved via activation through a combination of DMSO and TFAA.

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