ChemInform Abstract: A Simple Approach to β-Amino Acids by Acylation of Arenes with N-Acyl Aspartic Anhydrides.

✍ Scribed by A. G. GRIESBECK; H. HECKROTH

• Publisher: John Wiley and Sons
• Year: 2010
• Weight: 35 KB
• Volume: 29
• Category: Article
• ISSN: 0931-7597
• DOI: 10.1002/chin.199810221

✦ Synopsis

A Simple Approach to β-Amino Acids by Acylation of Arenes with N-Acyl Aspartic Anhydrides.

-Friedel-Crafts acylation of arenes with aspartic anhydrides generates a mixture of α-and β-amino acids. The highest β-selectivities are found for educt (Va).

-(GRIESBECK, A. G.;