A short and unequivocal synthesis of 5-a
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Edith Bencteux; Raymond Houssin
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Article
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1997
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Journal of Heterocyclic Chemistry
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English
β 272 KB
## Abstract The discovery of 4β(3βbromoanilino)β6,7βdimethoxyquinazoline (PD 153035) as an extremely potent inhibitor of the tyrosine kinase activity of the epidermal growth factor receptor led to the preparation of several fused tricyclic quinazoline analogues. The present paper reports a new tric