ChemInform Abstract: A Concise Preparation of 4-Borono-L-phenylalanine (L-BPA) from L-Phenylalanine.

✍ Scribed by Christophe Malan; Christophe Morin

• Publisher: John Wiley and Sons
• Year: 2010
• Weight: 27 KB
• Volume: 30
• Category: Article
• ISSN: 0931-7597
• DOI: 10.1002/chin.199912208

✦ Synopsis

A Concise Preparation of 4-Borono-L-phenylalanine (L-BPA) from L-Phenylalanine.

-The title compound (III), an important member of the family of boronated analogues of biomolecules, is conveniently prepared by Pd-catalyzed coupling of the N-protected iodophenylalanine derivative (I) with diboronate and following deprotection.

-(MALAN, CHRISTOPHE;