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ChemInform Abstract: 2,2-Dicyanovinyl as a Nonaromatic Aryl Bioisostere: Synthesis, Binding Experiments, and SAR Studies of Highly Selective Dopamine D4 Receptor Ligands.

✍ Scribed by Christian Haubmann; Harald Huebner; Peter Gmeiner


Publisher
John Wiley and Sons
Year
2010
Weight
30 KB
Volume
30
Category
Article
ISSN
0931-7597

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✦ Synopsis


2,2-Dicyanovinyl as a Nonaromatic Aryl Bioisostere: Synthesis, Binding Experiments, and SAR Studies of Highly Selective Dopamine D4 Receptor Ligands. -Title compounds of type (I) are tested for their dopamine receptor binding activity. Both types of 4-or 5-substituted compounds show selective dopamine D 4 receptor affinity. -(HAUBMANN,