𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Chemical synthesis of hormone receptor probes: high affinity photoactivated enediyne-estrogens

✍ Scribed by Ajay Purohit; Justin Wyatt; George Hynd; Justin Wright; Ahmed El-Shafey; Narashima Swamy; Rahul Ray; Graham B Jones


Book ID
104231947
Publisher
Elsevier Science
Year
2001
Tongue
French
Weight
88 KB
Volume
42
Category
Article
ISSN
0040-4039

No coin nor oath required. For personal study only.


📜 SIMILAR VOLUMES


A chemical probe for the estrogen recept
✍ Jeffrey A. Dodge; Mark G. Stocksdale; C. David Jones 📂 Article 📅 1995 🏛 John Wiley and Sons 🌐 French ⚖ 360 KB

## Abstract Radiolabelled raloxifene (LY156758) has been prepared by tritium gas hydrogenolysis of a 3‐aroyl‐__bis__‐brominated precursor. The requisite halogenated intermediate was accessed by regioselective aroylation of benzothiophene 6 with the acid chloride of 3,5‐dibromo‐4‐[2‐(1‐piperdinyl)et