Characterization of antagonistic activit
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Yoshihisa Ito; Tamami Koshiba; Masayo Doi; Satoru Asami; Hideomi Fukuda; Yoshie
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Article
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1992
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John Wiley and Sons
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English
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Experiments were performed to characterize the antagonistic activity and binding properties of SR 95531 [2-(3'carbethoxy-2'-propyl)-3-amino-6-paramethoxyphenyl-piridazinium bromide] in rat brain. SR 95531 and bicuculline methiodide inhibited muscimol-stimulated 36Cl-uptake in cortical synaptoneuroso