✦ LIBER ✦

Cariprazine (RGH-188), a potent D3/D2 dopamine receptor partial agonist, binds to dopamine D3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

✍ Scribed by István Gyertyán; Béla Kiss; Katalin Sághy; Judit Laszy; Györgyi Szabó; Tamás Szabados; Larisza I. Gémesi; Gabriella Pásztor; Mária Zájer-Balázs; Margit Kapás; Éva Ágai Csongor; György Domány; Károly Tihanyi; Zsolt Szombathelyi

Book ID: 116765732
Publisher: Elsevier Science
Year: 2011
Tongue: English
Weight: 897 KB
Volume: 59
Category: Article
ISSN: 0197-0186
DOI: 10.1016/j.neuint.2011.07.002

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

P.3.c.053 Dopamine D2/D3 receptor occupa

P.3.c.053 Dopamine D2/D3 receptor occupancy of RGH-188, a D3/D2 antagonist/partial agonist antipsychotic, in healthy volunteers

✍ I. Laszlovszky; G. N´emeth; G. P´asztor M´esz´aros; M. Kap´as; D.J. Brooks; N. P 📂 Article 📅 2007 🏛 Elsevier Science 🌐 English ⚖ 60 KB

P.3.d.015 Pharmacokinetics of RGH-188, a

P.3.d.015 Pharmacokinetics of RGH-188, a novel dopamine D3/D2 antagonist/partial agonist atypical antipsychotic, in rats and dogs

✍ G. Pásztor Mészáros; E. Terjéki Bolf; L. Gémesi; M. Kapáas; K. Tihanyi; Z. Szomb 📂 Article 📅 2008 🏛 Elsevier Science 🌐 English ⚖ 68 KB

P.3.d.007 F15063, a novel antipsychotic

P.3.d.007 F15063, a novel antipsychotic with dopamine D2/D3 antagonist, 5-HT1A agonist and D4 partial agonist properties: III. Duration of brain D2-like receptor occupancy, antipsychotic-like activity and plasma concentration in rodents

✍ M.B. Assié; L. Bardin; A.L. Auclair; N. Consul-Denjean; F. Sautel; M.S. Kleven; 📂 Article 📅 2006 🏛 Elsevier Science 🌐 English ⚖ 63 KB

The in vivo effects of olanzapine and ot

The in vivo effects of olanzapine and other antipsychotic agents on receptor occupancy and antagonism of dopamine D1, D2, D3, 5HT2A and muscarinic receptors

✍ W. Zhang; F. P. Bymaster 📂 Article 📅 1999 🏛 Springer 🌐 English ⚖ 172 KB

F15063, a potential antipsychotic with d

F15063, a potential antipsychotic with dopamine D2/D3antagonist, 5-HT1Aagonist and D4partial agonist properties: (IV) duration of brain D2-like receptor occupancy and antipsychotic-like activity versus plasma concentration in mice

✍ Marie-Bernadette Assié; Laurent Bardin; Agnès Auclair; Nathalie Consul-Denjean; 📂 Article 📅 2007 🏛 Springer-Verlag 🌐 English ⚖ 227 KB

Blockade of in vivo binding of 125I-labe

Blockade of in vivo binding of 125I-labeled 3-iodobenzamide (IBZM) to dopamine receptors by D2 antagonist and agonist

✍ W. Singhaniyom; Y.F. Tsai; T. Brücke; C.A. McLellan; R.M. Cohen; H.F. Kung; C.C. 📂 Article 📅 1988 🏛 Elsevier Science 🌐 English ⚖ 348 KB