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Biotransformation of Ergot Alkaloids by Haloperoxidase fromStreptomyces aureofaciens: Stereoselective Acetoxylation and Propionoxylation

✍ Scribed by Křen, Vladimír ;Kawuloková, Libuše ;Sedmera, Petr ;Polášek, Miroslav ;Lindhorst, Thisbe K. ;van Pée, Karl-Heinz


Book ID
102902610
Publisher
John Wiley and Sons
Year
1997
Tongue
English
Weight
516 KB
Volume
1997
Category
Article
ISSN
0947-3440

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✦ Synopsis


I Enzyme catalysis I Oxidases I Peroxides I Acylations Agroclavine (1) was oxidized, by haloperoxidase from Strep-2,3-dihydro-6,8-dimethyl-3~-propionoxy-8-ergolen-2-one (4). tomyces aureofaciens, to 2,3-dihydro-6,8-dimethyl-3P-ace-The biotransformation proceeded faster in the propionate toxy-8-ergolen-2-one (2) in the presence of sodium acetate buffer, affording also the higher oxidation product and bromine ions. Acetate was incorporated into the above (4aS),( 10bS)-7-amino-3,4,4a,5,6,lOb-hexahydro-2,4-dimeth- product during oxidation. In a propionate buffer, incorporayl-6-oxobenzo(f]quinoline (3). tion of propionate into the product was observed, yielding