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Binding characteristics of the glucocorticoid receptor in peripheral blood lymphocytes in multiple sclerosis

✍ Scribed by Florian Then Bergh; Annette Grasser; Claudia Trenkwalder; Herbert Backmund; Florian Holsboer; Rainer Rupprecht


Publisher
Springer
Year
1999
Tongue
English
Weight
93 KB
Volume
246
Category
Article
ISSN
0340-5354

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Benzodiazepine (BDZ) binding sites were studied by using 3H-diazepam and 3H-Ro 5-4864 in intact lymphocytes from peripheral blood (PBL), in comparison to kidney and cerebellum. Experiments with 3H-diazepam performed at equilibrium and measuring kinetics revealed that BDZ binding sites are indeed pre