The synthesis of chiral annulet 1,4,7-tr
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Gilles Argouarch; Colin L Gibson; Graham Stones; David C Sherrington
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Article
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2002
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Elsevier Science
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French
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Novel and flexible routes for the synthesis of chiral ring annulet 2,6-disubstituted 1,4,7-trimethyl-1,4,7-triazamacrocycles are described. Efficient macrocyclisations were realised provided that chiral analogues of N,N-bis-[2-(toluene-sulfonylamino)ethyl]-toluene-4-sulfonamide were used as the nucl