✦ LIBER ✦

Azole Endothelin Antagonists. 2. Structure−Activity Studies

✍ Scribed by von Geldern, Thomas W.; Kester, Jeffrey A.; Bal, Radhika; Wu-Wong, Jinshyun R.; Chiou, William; Dixon, Douglas B.; Opgenorth, Terry J.

Book ID: 121313851
Publisher: American Chemical Society
Year: 1996
Tongue: English
Weight: 380 KB
Volume: 39
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm950592+

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

ChemInform Abstract: Azole Endothelin An

ChemInform Abstract: Azole Endothelin Antagonists. Part 2. Structure-Activity Studies.

✍ T. W. VON GELDERN; J. A. KESTER; R. BAL; J. R. WU-WONG; W. CHIOU; D. B. DIXON; T 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 28 KB

Azole Endothelin Antagonists. 1. A Recep

Azole Endothelin Antagonists. 1. A Receptor Model Explains an Unusual Structure−Activity Profile

✍ von Geldern, Thomas W.; Hutchins, Charles; Kester, Jeffrey A.; Wu-Wong, Jinshyun 📂 Article 📅 1996 🏛 American Chemical Society 🌐 English ⚖ 334 KB

ChemInform Abstract: Azole Endothelin An

ChemInform Abstract: Azole Endothelin Antagonists. Part 1. A Receptor Model Explains an Unusual Structure-Activity Profile.

✍ T. W. VON GELDERN; C. HUTCHINS; J. A. KESTER; J. R. WU-WONG; W. CHIOU; D. B. DIX 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 31 KB

Design and Structure--Activity Relations

Design and Structure--Activity Relationship of Novel Endothelin Receptor A Tripeptide Antagonists

✍ Junjun Dong; Ning Yang; Yuanjun Liang; Ping Wu; Xin Li; Keliang Liu 📂 Article 📅 2005 🏛 Springer Netherlands 🌐 English ⚖ 227 KB

Structure–activity relationship studies

Structure–activity relationship studies on 2-heteroaryl-4-arylimidazoles NPY5 receptor antagonists

✍ Richard L. Elliott; Robert M. Oliver; Janet A. LaFlamme; Melissa L. Gillaspy; Ma 📂 Article 📅 2003 🏛 Elsevier Science 🌐 English ⚖ 142 KB

A series of 2-heteroaryl-4-arylimidazoles with potent in vitro activity at the NPY5 receptor was developed. Introduction of electron-withdrawing groups on the 4-aryl ring led to a significant improvement of in vitro potency. Several analogues from this series had anorectic activity in rodent feeding

Structure—Activity Relationship Studies

Structure—Activity Relationship Studies on 2-Heteroaryl-4-arylimidazoles NPY5 Receptor Antagonists.

✍ Richard L. Elliott; et al. et al. 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 67 KB 👁 1 views