𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Aza-annulation as a route to hydroxylated alkaloid lipids. The synthesis of (±)-prosopinine

✍ Scribed by Gregory R. Cook; Lars G. Beholz; John R. Stille

Publisher
Elsevier Science
Year
1994
Tongue
French
Weight
300 KB
Volume
35
Category
Article
ISSN
0040-4039

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

The aza-robinson annulation: An applicat
The aza-robinson annulation: An application to the synthesis of iso-A58365A
✍ Francis G. Fang; Maurizio Prato; Guncheol Kim; Samuel J. Danishefsky 📂 Article 📅 1989 🏛 Elsevier Science 🌐 French ⚖ 258 KB

Annulation of diazomethylvinylketone (4a) with a variety of secondary thiolactams provides a novel route to dihydro-y-pyridones. This approach has been applied to the synthesis of iso-A58365A ( ), the y-pyridone analog of the ACE inhibitor, A58365A (1). We have recently described a novel route to

Aza-annulation as a versatile approach t
Aza-annulation as a versatile approach to the synthesis of non-benzodiazepene compounds for the treatment of sleep disorders
✍ Petr Benovsky; John R Stille 📂 Article 📅 1997 🏛 Elsevier Science 🌐 French ⚖ 233 KB

The aza-annulation of enamino ester substrates has been demonstrated as an efficient alternative to the syntheses of non-benzodiazepine sleep inducers. Enamino ester substrates derived from aryl, thiophene, and indole functionality were prepared from the corresponding ethyl amines by isothiocyanate