Asymmetric synthesis of aziridine 2-phos
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Franklin A. Davis; William McCoull
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Article
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1999
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Elsevier Science
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French
⚖ 266 KB
Enantiopure sulfinimine (S)-4 was employed in a Darzens-type synthesis of aziridine 2-phosphonates (-)-7/(+)-8 which were transformed into a-amino phosphonates (S)-11/(R)-12 and the first enantiopure examples of azirinyl phosphonates 13-15.