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Application of a new amidophosphite ligand to Rh-catalyzed asymmetric hydrogenation of β-dehydroamino acid derivatives in supercritical carbon dioxide: Activation effect of protic co-solvents

✍ Scribed by Sergey E. Lyubimov; Eugenie A. Rastorguev; Vadim A. Davankov


Publisher
John Wiley and Sons
Year
2011
Tongue
English
Weight
95 KB
Volume
23
Category
Article
ISSN
0899-0042

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✦ Synopsis


Abstract

New chiral amidophosphite ligand was synthesized and tested in the Rh‐catalyzed asymmetric hydrogenation of (Z)‐β‐(acylamino)acrylates in protic solvents and supercritical carbon dioxide (scCO~2~) The catalytic performance is affected greatly by the acidity of the solvents. Better enantioselectivity (up to 88% ee) was achieved in scCO~2~ containing 1,1,1,3,3,3‐hexafluoro‐2‐propanol, compared to neat protic solvents. Chirality, 2011. © 2011 Wiley‐Liss, Inc.