✦ LIBER ✦

Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 1: Discovery and SAR study of 4-pyrazolylpiperidine side chains

✍ Scribed by Dong-Ming Shen; Min Shu; Sander G. Mills; Kevin T. Chapman; Lorraine Malkowitz; Martin S. Springer; Sandra L. Gould; Julie A. DeMartino; Salvatore J. Siciliano; Gloria Y. Kwei; Anthony Carella; Gwen Carver; Karen Holmes; William A. Schleif; Renee Danzeisen; Daria Hazuda; Joseph Kessler; Janet Lineberger; Michael D. Miller; Emilio A. Emini

Book ID: 108073184
Publisher: Elsevier Science
Year: 2004
Tongue: English
Weight: 233 KB
Volume: 14
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2003.12.004

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Antagonists of Human CCR5 Receptor Conta

Antagonists of Human CCR5 Receptor Containing 4-(Pyrazolyl)piperidine Side Chains. Part 1. Discovery and SAR Study of 4-Pyrazolylpiperidine Side Chains.

✍ Dong-Ming Shen; et al. et al. 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 168 KB 👁 2 views

Antagonists of Human CCR5 Receptor Conta

Antagonists of Human CCR5 Receptor Containing 4-(Pyrazolyl)piperidine Side Chains. Part 3. SAR Studies on the Benzylpyrazole Segment.

✍ Min Shu; et al. et al. 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 123 KB 👁 2 views

Antagonists of Human CCR5 Receptor Conta

Antagonists of Human CCR5 Receptor Containing 4-(Pyrazolyl)piperidine Side Chains. Part 2. Discovery of Potent Selective, and Orally Bioavailable Compounds.

✍ Dong-Ming Shen; et al. et al. 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 65 KB 👁 2 views

## Abstract For Abstract see ChemInform Abstract in Full Text.

Antagonists of human CCR5 receptor conta

Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 2: Discovery of potent, selective, and orally bioavailable compounds

✍ Dong-Ming Shen; Min Shu; Christopher A. Willoughby; Shrenik Shah; Christopher L. 📂 Article 📅 2004 🏛 Elsevier Science 🌐 English ⚖ 218 KB

1,3,4-Trisubstituted Pyrrolidine CCR5 Re

1,3,4-Trisubstituted Pyrrolidine CCR5 Receptor Antagonists: Modifications of Arylpropylpiperidine Side Chains.

✍ Christopher L. Lynch; et al. et al. 📂 Article 📅 2003 🏛 John Wiley and Sons ⚖ 12 KB 👁 1 views

Synthesis and SAR Studies of 4-(Heteroar

Synthesis and SAR Studies of 4-(Heteroarylpiperidin-1-yl-methyl)-pyrrolidin-1-yl-acetic Acid Antagonists of the Human CCR5 Chemokine Receptor.

✍ K. Shankaran; et al. et al. 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 16 KB 👁 2 views