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Antagonist activity of novel angiotensin analogues substituted in positions 1, 5 and 8

✍ Scribed by Szalay, Ksz; Nyéki, O; Kisfaludy, L; Kárpáti, E; Szporny, L; Makara, Gb; Varga, B

Book ID: 122831679
Publisher: Elsevier Science
Year: 1985
Tongue: English
Weight: 57 KB
Volume: 13
Category: Article
ISSN: 0167-0115
DOI: 10.1016/0167-0115(85)90100-4

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## Abstract A sterically constrained non‐coded amino acid, 1‐aminocyclopentane‐1‐carboxylic acid (Apc), was introduced in position 7 or 8 of the bradykinin (BK) B~2~ receptor antagonist, [D‐Arg^0^, Hyp^3^, Thi^5, 8^, D‐Phe^7^]BK, previously synthesized by Stewart's group. This modification is belie