An improved synthesis of solid-supported reagents (SSRs) for selective acylation of amines by microwave irradiation

✍ Scribed by Elena Petricci; Maurizio Botta; Federico Corelli; Claudia Mugnaini

• Book ID: 104251812
• Publisher: Elsevier Science
• Year: 2002
• Tongue: French
• Weight: 150 KB
• Volume: 43
• Category: Article
• ISSN: 0040-4039
• DOI: 10.1016/s0040-4039(02)01478-8

✦ Synopsis

Microwave-assisted acylation of a solid-supported pyrimidine linker with different acyl chlorides gave polymer-bound 4-acyloxypyrimidines, which in turn were used as SSRs for rapid and selective acylation of amines under microwave irradiation.