An Efficient Synthesis of 5-(or 6-)Arylbenzoindolizidine and -quinolizidine Derivatives

✍ Scribed by Stéphane Lebrun; Axel Couture; Eric Deniau; Pierre Grandclaudon

• Publisher: John Wiley and Sons
• Year: 1999
• Tongue: English
• Weight: 236 KB
• Volume: 1999
• Category: Article
• ISSN: 1434-193X
• DOI: 10.1002/(sici)1099-0690(199909)1999:9<2345::aid-ejoc2345>3.0.co;2-p

✦ Synopsis

A new methodology for the synthesis of (hetero)arylated based aromatic enamides, and ultimate cyclization, is reported. benzoindolizidine and benzoquinolizidine derivatives through sequential reduction of pyrrolidine-and piperidine- [a]