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An Efficient, Direct Bis-ortho-chlorination of 4-(Difluoromethoxy)aniline and Its Application to the Synthesis of BMS-665053, a Potent and Selective Pyrazinone-Containing Corticotropin-Releasing Factor-1 Receptor Antagonist

✍ Scribed by Li, Jianqing; Smith, Daniel; Krishnananthan, Subramaniam; Hartz, Richard A.; Dasgupta, Bireshwar; Ahuja, Vijay; Schmitz, William D.; Bronson, Joanne J.; Mathur, Arvind; Barrish, Joel C.; Chen, Bang-Chi


Book ID
120252199
Publisher
American Chemical Society
Year
2012
Tongue
English
Weight
303 KB
Volume
16
Category
Article
ISSN
1083-6160

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