✦ LIBER ✦

Allosteric Control of Ligand Selectivity between Estrogen Receptors α and β: Implications for Other Nuclear Receptors

✍ Scribed by Kendall W. Nettles; Jun Sun; James T. Radek; Shubin Sheng; Alice L. Rodriguez; John A. Katzenellenbogen; Benita S. Katzenellenbogen; Geoffrey L. Greene

Book ID: 117737351
Publisher: Elsevier Science
Year: 2004
Tongue: English
Weight: 705 KB
Volume: 13
Category: Article
ISSN: 1097-2765
DOI: 10.1016/s1097-2765(04)00054-1

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

A Ligand-Based Approach to Understanding

A Ligand-Based Approach to Understanding Selectivity of Nuclear Hormone Receptors PXR, CAR, FXR, LXRα, and LXRβ

✍ Sean Ekins; Leonid Mirny; Erin G. Schuetz 📂 Article 📅 2002 🏛 Springer US 🌐 English ⚖ 747 KB

Selectivity of antibodies to estrogen re

Selectivity of antibodies to estrogen receptors α and β (ERα and ERβ) for detecting DNA-bound ERα and ERβ in vitro

✍ Valentyn V. Tyulmenkov; Carolyn M. Klinge 📂 Article 📅 2000 🏛 Elsevier Science 🌐 English ⚖ 194 KB

Structural Basis of Allosteric Ligand–Re

Structural Basis of Allosteric Ligand–Receptor Interactions in the Insulin/Relaxin Peptide Family : Implications for Other Receptor Tyrosine Kinases and G-Protein-Coupled Receptors

✍ Pierre De Meyts; Lisbeth Gauguin; Angela Manegold Svendsen; Mazen Sarhan; Louise 📂 Article 📅 2009 🏛 John Wiley and Sons 🌐 English ⚖ 243 KB

Synthesis and Biological Evaluation of a

Synthesis and Biological Evaluation of a Novel Series of Furans: Ligands Selective for Estrogen Receptor α

✍ Mortensen, Deborah S.; Rodriguez, Alice L.; Carlson, Kathryn E.; Sun, Jun; Katze 📂 Article 📅 2001 🏛 American Chemical Society 🌐 English ⚖ 293 KB

Identification of heme as the ligand for

Identification of heme as the ligand for the orphan nuclear receptors REV-ERBα and REV-ERBβ

✍ Raghuram, Srilatha; Stayrook, Keith R; Huang, Pengxiang; Rogers, Pamela M; Nosie 📂 Article 📅 2007 🏛 Nature Publishing Group 🌐 English ⚖ 454 KB

Rational Design of Highly Active and Sel

Rational Design of Highly Active and Selective Ligands for the α5β1 Integrin Receptor

✍ Dominik Heckmann; Axel Meyer; Burkhardt Laufer; Grit Zahn; Roland Stragies; Hors 📂 Article 📅 2008 🏛 John Wiley and Sons 🌐 English ⚖ 735 KB

## Abstract The inhibition of integrin function is a major challenge in medicinal chemistry. Potent ligands are currently in different stages of clinical trials for the antiangiogenic therapy of cancer and age‐related macula degeneration (AMD). The subtype α5β1 has recently been drawn into the focu