Synthesis and evaluation of derivatives
✍
Heekyung Choi; Thomas F. Murray; Jane V. Aldrich
📂
Article
📅
2003
🏛
Wiley (John Wiley & Sons)
🌐
English
⚖ 82 KB
As part of an effort to develop peptide-based affinity labels for opioid receptors, [Leu(5)]enkephalin (LeuEnk) and DTLET (Tyr-D-Thr-Gly-Phe-Leu-Thr), potent agonists for delta receptors, were selected as the parent peptides for further modification. The affinity label derivatives were prepared usin