threo-a-Dibensylamino-B-hydroxyesters (2) have been synthesised with high diastereoselectivity through the NaBH reduction of a-dibenzylamino-B-oxoesters (4) and then tranformed into threo-a-amino-B-hydroxyac?ds. a-Amino-B-hydroxyacids are derivatives of primary importance both as enzymatic inhibito
Acid catalysis in aldol condensation of α-amino silyl ketene acetals. Diastereoselective synthesis of α-amino-β-hydroxyacids.
✍ Scribed by Giuseppe Guanti; Luca Banfi; Enrica Narisano; Carlo Scolastico
- Publisher
- Elsevier Science
- Year
- 1985
- Tongue
- French
- Weight
- 217 KB
- Volume
- 26
- Category
- Article
- ISSN
- 0040-4039
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