ChemInform Abstract: Synthesis of 3-Hydr
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M. SUNOSE; K. M. ANDERSON; A. G. ORPEN; T. GALLAGHER; S. J. F. MACDONALD
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Article
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2010
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John Wiley and Sons
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Synthesis of 3-Hydroxy and 3-Amino 2-Substituted N-Heterocycles via Enamine Oxidation and Aziridination. -Usual asymmetric epoxidation of the N-sulfonyl heterocyclic enamines (I) followed by methanolysis results in formation of 2,3-dihydroxy derivatives. Only diol derivatives are also obtained unde