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A simplified synthesis of 18F-labelled cytosine- and uracil-nucleosides

✍ Scribed by Gerard W.M. Visser; Paul Noordhuis; Oene Zwaagstra; Jacobus D.M. Herscheid; Arend Hoekstra

Publisher
Elsevier Science
Year
1986
Weight
170 KB
Volume
37
Category
Article
ISSN
0883-2889

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✦ Synopsis

tSF-labelled cytosine-and uracil-nucleosides are synthesized starting from their unprotected parent nucleosides by reaction with acetylhypofluorite in acetic acid in an overall radiochemical yield of 20 and 30% respectively.

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