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A Physiologically Based Pharmacokinetic Analysis of Capecitabine, a Triple Prodrug of 5-FU, in Humans: The Mechanism for Tumor-Selective Accumulation of 5-FU

✍ Scribed by Yuko Tsukamoto; Yukio Kato; Masako Ura; Ikuo Horii; Hideo Ishitsuka; Hiroyuki Kusuhara; Yuichi Sugiyama


Book ID
110295840
Publisher
Springer US
Year
2001
Tongue
English
Weight
372 KB
Volume
18
Category
Article
ISSN
0724-8741

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## Abstract The nonlinear pharmacokinetics of capecitabine, a triple prodrug of 5‐FU preferentially activated in tumour tissues, was investigated in human cancer xenograft models. A physiologically based pharmacokinetic (PBPK) model integrating the activation process of capecitabine to 5‐FU and 5‐F