An autoxidative approach to 1,2,3,4-tetr
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Michèle Bois-Choussy; Michaël De Paolis; Jieping Zhu
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Article
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2001
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Elsevier Science
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French
β 70 KB
Treatment of N-benzyl 1,2,3,4-tetrahydroisoquinoline-1-carboxylate with sodium hydride in N,N-dimethylformamide gives the corresponding N-benzyl 1,2,3,4-tetrahydroisoquinolin-1-one in quantitative yield. The N-benzyl 1,2,3,4-tetrahydro-b-carbolin-1-one is prepared in a similar fashion. The N-deprote