A new entry to pyrazolo[4,3-e][1,4]diazepines. Facile synthesis of pyrazolo [4,3-e][1,4]diazepin-5,8-diones, 5,6,8-triones and pyrazolo[4,3-e]pyrrolo-[1,2-a][1,4]diazepin-5,10-diones
β Scribed by Nalla Ram Reddy; Ghanta Mahesh Reddy; Padi Pratap Reddy
- Publisher
- Journal of Heterocyclic Chemistry
- Year
- 2005
- Tongue
- English
- Weight
- 74 KB
- Volume
- 42
- Category
- Article
- ISSN
- 0022-152X
No coin nor oath required. For personal study only.
β¦ Synopsis
A facile approach to pyrazolo [4,3-e][1,4] diazepin-5,8-diones andpyrazolo[4,3-e]pyrrolo[1,2-a][1,4]diazepin-5,10-diones is reported. Strategy involved the utility of Ξ±-amino acid as a three-atom segment in the construction of diazepine skeleton on the preformed pyrazole ring.
π SIMILAR VOLUMES
## Abstract Fused tricyclic 7βphenylβ5__H__βthizolo[5,4β__e__]pyrrolo[1,2β__a__][1,4]diazepinβ10(9__H__)one (**10**) was prepared by thermolysis of 2βphenylβ4β(1βpyrrolylmethyl)thiazoleβ5βcarbonyl azide (**9**) in acetic acid. In addition, starting from **10**, 7βphenylβ5__H__βthiazolo [5,4β__e__][