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A highly effective method for synthesis of Nω-substituted arginines as building blocks for Boc/Fmoc peptide chemistry

✍ Scribed by Zoltán Székely; Sotir Zakhariev; Corrado Guarnaccia; Nikolinka Antcheva; Sándor Pongor

Book ID: 104261550
Publisher: Elsevier Science
Year: 1999
Tongue: French
Weight: 270 KB
Volume: 40
Category: Article
ISSN: 0040-4039
DOI: 10.1016/s0040-4039(99)00767-4

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✦ Synopsis

Chemically and optically pure N~-substituted arginine derivatives were prepared with high yields in two steps, starting from N%proteeted ornithine and ArSOzN=C(SMe)2. The compounds were applied to solid phase peptide synthesis using Boc as well as Fmoc chemistries.

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