𝔖 Bobbio Scriptorium
✦   LIBER   ✦

A general, one-pot method for the synthesis of 2-substituted oxazoles

✍ Scribed by Eric L. Williams

Publisher
Elsevier Science
Year
1992
Tongue
French
Weight
238 KB
Volume
33
Category
Article
ISSN
0040-4039

No coin nor oath required. For personal study only.

✦ Synopsis

The reaction of 2-irimcihylsilyi-1,2,3-triazole with acid chlorides readily forms iriazuie amides. The wiazole amides, when heated 10 15oOC in suifolane. rearrange wirh rhe elimination of niwngen to give 2-subslituied nxazoles in high yields. The nxazoie synlhesis is general. and can be carried 01~1 in one-pot.

πŸ“œ SIMILAR VOLUMES

A facile one-pot synthesis of 2,5-disubs
A facile one-pot synthesis of 2,5-disubstituted oxazoles using iodobenzene diacetate
✍ Rajender S. Varma; Dalip Kumar πŸ“‚ Article πŸ“… 1998 πŸ› Journal of Heterocyclic Chemistry 🌐 English βš– 150 KB πŸ‘ 1 views

## Abstract A facile one‐pot synthesis of oxazoles 1a‐h is described that utilizes readily available aromatic α‐methyl ketones and a safe hypervalent iodine reagent, iodobenzene diacetate.

A novel, general, totally stereoselectiv
A novel, general, totally stereoselective one-pot synthesis of cis-3-substituted 4-formylazetidin-2-ones
✍ Benito Alcaide; Yolanda MartΓ­n-Cantalejo; JoaquΓ­n Plumet; JuliΓ‘n RodrΓ­guez-LΓ³pez πŸ“‚ Article πŸ“… 1991 πŸ› Elsevier Science 🌐 French βš– 275 KB

## A general , totally stereoselectrve one-pot synthesis of cls-3-substttuted-+formylazetrdtn-2-ones based upon the reacuon of actd chlorides and 1,4-b~s-(4-methoxyphenyl)-I,4-drazabuta-IJ-d~ene, as synthettc equrvalent of the correspondmg unknown a-formyhmtne, has been developed Appropnately as-s