A Cyclic CCK8 Analogue Selective for the Cholecystokinin Type A Receptor: Design, Synthesis, NMR Structure and Binding Measurements

Cover Picture: A Cyclic CCK8 Analogue Se

Cover Picture: A Cyclic CCK8 Analogue Selective for the Cholecystokinin Type A Receptor: Design, Synthesis, NMR Structure and Binding Measurements (ChemBioChem 11/2003)

✍ Stefania De Luca; Raffaele Ragone; Chiara Bracco; Giuseppe Digilio; Luigi Aloj; 📂 Article 📅 2003 🏛 John Wiley and Sons 🌐 English ⚖ 21 KB

## Abstract **The cover picture shows** a molecular model of the interaction between the new CCK8 analogue, Cycle29,34[Dpr29,Lys34]‐CCK8 (shown as a CPK model) and the receptor fragment CCK~A~‐R(1–47) (represented by a pink ribbon). The introduction of the cyclic constraint between the Dpr29 sidech